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Inhibitors
5-HT Receptor Inhibitors
1
AAK1 Inhibitors
6
ACC1 Inhibitors
1
ACE Inhibitors
45
Acyltransferase Inhibitors
3
AICARFT Inhibitors
2
AIMP2-DX2 Inhibitors
2
AKT Inhibitors
12
Aldose Reductase Inhibitors
9
ALK Inhibitors
14
ALK-BET Inhibitors
1
Allosteric Inhibitors
3
AMCase Inhibitors
2
Aminopeptidase Inhibitors
2
Aromatase Inhibitors
5
AS Inhibitors
3
ATAD2 Inhibitors
1
ATM Kinase Inhibitors
2
ATP Synthase Inhibitors
3
ATR Inhibitors
1
Aurora Kinase Inhibitors
18
Autophagy Inhibitors
2
Autotaxin Inhibitors
1
AXL Inhibitors
3
BACE Inhibitors
15
BCL Inhibitors
3
BCR-ABL Inhibitors
8
BET Inhibitors
33
beta-Lactamase Inhibitors
27
BRAF Inhibitors
3
BRM Inhibitors
0
BTK Inhibitors
16
c-KIT Inhibitors
3
c-Met Inhibitors
2
CA Inhibitors
14
Calpain Inhibitors
1
Cathepsin C Inhibitors
3
Cathepsin K Inhibitors
3
CD38 Inhibitors
2
CD73 Inhibitors
2
CDK Inhibitors
23
CEN Inhibitors
2
CETP Inhibitors
1
CHK1 Inhibitors
6
CK Inhibitors
1
COMT Inhibitors
1
COX Inhibitors
8
CRK12 Inhibitors
1
CSF-1R Inhibitors
5
CY P450 Inhibitors
1
DAGL Inhibitors
3
DcpS Inhibitors
1
DGAT1 Inhibitors
1
DHFR Inhibitors
4
DHODH Inhibitors
5
DLK-MAP Kinase Inhibitors
1
DNA Gyrase Inhibitors
3
DNA Polymerase Inhibitors
4
DNA-PK Inhibitors
3
DPP-4 Inhibitors
12
DPP1 Inhibitors
1
DprE1 Inhibitors
6
DYRK Inhibitors
2
EED Inhibitors
1
EGFR Inhibitors
29
EL Inhibitors
2
Ergosterol Inhibitors
1
ERK Inhibitors
16
EZH2 Inhibitors
2
FAAH Inhibitors
1
FABP Inhibitors
3
Factor D Inhibitors
2
Factor VIIa Inhibitors
1
Factor Xa Inhibitors
5
Factor XIa Inhibitors
5
FAK Inhibitors
1
FDP Inhibitors
2
FGFR Inhibitors
9
FLAP Inhibitors
9
FLT Inhibitors
3
Fyn Kinase Inhibitors
2
GAK Inhibitors
1
Glutaminase Inhibitors
1
Glycine Transporter-1 Inhibitors
1
GRK2 Inhibitors
2
GSK-3 Inhibitors
5
GST Inhibitors
1
HAT Inhibitors
2
HBV Capsid Inhibitors
1
HCV Inhibitors
6
HDAC Inhibitors
7
Hedgehog Inhibitors
1
HIF Inhibitors
3
HIV Inhibitors
4
HIV-1 Inhibitors
3
HMT Inhibitors
3
HNE Inhibitors
1
HSD1 Inhibitors
1
hSERT Inhibitors
4
Hsp90 Inhibitors
16
HSV Inhibitors
1
Human Arginase Inhibitors
2
Hydroxylase Inhibitors
2
IBAT Inhibitors
1
IDH1 Inhibitors
11
IDH2 Inhibitors
2
IDO Inhibitors
15
IGF-1R Inhibitors
1
IKK Inhibitors
8
iNOS Inhibitors
8
Integrase Inhibitors
9
Integrin Inhibitors
3
IRAK4 Inhibitors
6
ITK Inhibitors
1
JAK Inhibitors
25
KDM Inhibitors
3
KEAP1-NRF2 Inhibitors
2
KHK Inhibitors
1
Kinesin Inhibitors
1
KMO Inhibitors
1
KRAS-G12C Inhibitors
7
L3MBTL3 Inhibitors
1
LDH Inhibitors
1
Lipase Inhibitors
1
LMP2 Inhibitors
1
LOX Inhibitors
6
LpxC Inhibitors
8
LRRK2 Inhibitors
1
LSD1 Inhibitors
1
MAGL Inhibitors
4
MAO-B Inhibitors
2
MAPK Inhibitors
21
MCHR1 Inhibitors
2
MCL-1 Inhibitors
10
MDM2 Inhibitors
3
MEK Inhibitors
15
Menin-MLL Inhibitors
9
MET Inhibitors
1
MetAP2 Inhibitors
1
MMP Inhibitors
5
MNK Inhibitors
3
mPGES-1 Inhibitors
2
MPO Inhibitors
2
MPS1 Inhibitors
2
Mps1 Kinase Inhibitors
7
MRTF/SRF Inhibitors
1
mTOR Inhibitors
22
MTP Inhibitors
2
NAMPT Inhibitors
2
NaV1.7 Inhibitors
8
NF-kB Inhibitors
9
NLRP3 Inhibitors
2
nNOS Inhibitors
2
NNRT Inhibitors
20
non-BET Inhibitors
0
non-Prostanoid Inhibitors
1
NOX Inhibitors
3
NRT Inhibitors
19
NS3/4A Inhibitors
8
NS4B Inhibitors
1
NS5A Inhibitors
10
NS5B Inhibitors
8
NSK Inhibitors
1
OAT Inhibitors
1
Other Targets
4
p97 Inhibitors
6
Pan-Aurora Inhibitors
2
Pan-JAK Inhibitors
1
Pan-KIT Mutant Inhibitors
1
Pan-Pim Inhibitors
3
Pan-RAF Inhibitors
2
Pan-TRK Inhibitors
4
Parasite Inhibitors
1
PARG Inhibitors
2
PARP Inhibitors
0
PD1-PD-L1 Inhibitors
3
PDE Inhibitors
6
PDE1 Inhibitors
1
PDE10A Inhibitors
2
PDE2 Inhibitors
3
PDE2A Inhibitors
5
PDE3 Inhibitors
2
PDE4 Inhibitors
15
PDE5 Inhibitors
5
PDGFR Inhibitors
9
PDHK Inhibitors
1
PERK Inhibitors
2
PfEF2 Inhibitors
2
PHGDH Inhibitors
2
PI3K Inhibitors
91
PI4K Inhibitors
2
PLA-2 Inhibitors
1
PLK1 Inhibitors
1
Porcupine Inhibitors
1
PP Inhibitors
1
Protease Inhibitors
16
Proteasome Inhibitors
8
Proton Pump Inhibitors
2
RAF Inhibitors
7
RET Inhibitors
5
RIP Inhibitors
13
ROCK Inhibitors
6
RORyt Inhibitors
2
ROS Inhibitors
4
RSV Fusion Inhibitors
13
RTK Inhibitors
10
SAHH Inhibitors
8
SARS-CoV Inhibitors
9
sEH Inhibitors
4
SERD Inhibitors
3
Serine Protease Inhibitors
2
SERT Inhibitors
2
sGC Inhibitors
1
SGLT1 Inhibitors
2
SGLT2 Inhibitors
5
SHP2 Inhibitors
4
SMO Inhibitors
4
SMYD Inhibitors
2
SphK2 Inhibitors
1
SPIN1 Inhibitors
1
SPPL2a inhibitors
1
Src Inhibitors
4
SSR Inhibitors
6
STAT Inhibitors
2
Syk Inhibitors
6
Tankyrase Inhibitors
5
TLR Inhibitors
7
TNF Inhibitors
2
Topo II Inhibitors
1
Topoisomerase Inhibitors
2
TPH Inhibitors
3
TRK Inhibitors
7
TRPV4 Inhibitors
3
TTK Inhibitors
5
TTR Amyloid Inhibitors
2
Tubulin Inhibitors
1
TYK Inhibitors
2
URAT1 Inhibitors
2
VEGFR Inhibitors
26
VMAT Inhibitors
2
WDR5 Inhibitors
1
XO Inhibitors
1
XOR Inhibitors
1
yGS Inhibitors
1
ZAK Inhibitors
1
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