9-Cyclopentyl-2-((2-ethoxy-4-(4-hydroxypiperidin-1-yl)phenyl)amino)-5-methyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one

SI-4107

9-Cyclopentyl-2-((2-ethoxy-4-(4-hydroxypiperidin-1-yl)phenyl)amino)-5-methyl-8,9-dihydro-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one, >98% (HPLC)

CAS No. : [1228817-38-6]

MDL No. : MFCD28167735

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Applications : A potent, selective and ATP-competitive dual Mps1/Plk1 inhibitor, with an IC₅₀ and a Kd of 145 nM and 12 nM for Mps1 and a Kd of 61 nM for Plk1.

References : Liu Y. et al.: J. Med. Chem., 58(8), 3366-3392, 2015.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.