A804598

SI-6170

A804598, >98% (HPLC)

CAS No. : [1125758-85-1]

IUPAC Name : (S,Z)-2-Cyano-1-(1-phenylethyl)-3-(quinolin-5-yl)guanidine

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
250MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
500MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : A804598 is a CNS‑penetrant, competitive P2X7 receptor antagonist that blocks mouse, rat, and human P2X7 channels with IC₅₀ values of 9–11 nM. Its potency and BBB permeability support its use in studies of P2X7‑driven inflammation and neurodegeneration.

References : Donnelly-Roberts D. L. et al.: Neuropharmacology, 56(1), 223-9, 2009; He Y. et al.: Neuroinflammation, 14(1),135, 2017; Fabbrizio P. et al.: Cell Neurosci., 11, 249, 2017.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.