ACK1 inhibitor

SI-7952

ACK1 inhibitor, >98% (HPLC)

IUPAC Name : 3-(8-Amino-1-(2-methoxy-4-phenoxyphenyl)imidazo[1,5-a]pyrazin-3-yl)-1-methylcyclobutan-1-ol

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
5MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
10MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : This compound emerged as a key early ACK1 lead, exhibiting cellular ACK1 inhibition with an IC₅₀ of 35 nM and showing favorable ADME properties, establishing it as a strong foundation for further optimization toward selective, drug‑like ACK1 inhibitors suitable for anticancer development.

References : Jin M. et al.: Bioorg. Med. Chem. Lett., 23(4), 979-984, 2013.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.