Alcaftadine

SI-4228

Alcaftadine, >98% (HPLC)

CAS No. : [147084-10-4]

MDL No. : MFCD09954106

Synonyms : Lastacaft; R89674

IUPAC Name : 11-(1-Methylpiperidin-4-ylidene)-6,11-dihydro-5H-benzo[d]imidazo[1,2-a]azepine-3-carbaldehyde

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
25MG	95.00		Back Order	Estimated to ship on 04 October 2026
50MG	125.00		Back Order	Estimated to ship on 04 October 2026
100MG	195.00		Back Order	Estimated to ship on 04 October 2026
250MG	295.00		Back Order	Estimated to ship on 04 October 2026
500MG	495.00		Back Order	Estimated to ship on 04 October 2026

Applications : Alcaftadine is a high affinity ligand for the H1 receptor, with a pKi (8.5) that is comparable with that of other H1 antihistamines. Alcaftadine is also an antagonist for H2 and H4 receptors with no affinity for the H3 receptor. It is used to prevent eye irritation and treat the signs and symptoms of allergic conjunctivitis.

References : Ding H. X. et al.: Bioorg. Med. Chem. 21(11), 2795-2825, 2013.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.