AM-1241

SI-7282

AM-1241, >98% (HPLC)

CAS No. : [444912-48-5]

Synonyms : (R,S)-3-(2-Iodo-5-nitrobenzoyl)-1-(1-methyl-2-piperidinylmethyl)-1H-indole

IUPAC Name : (2-Iodo-5-nitrophenyl)(1-((1-methylpiperidin-2-yl)methyl)-1H-indol-3-yl)methanone

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
5MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
10MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : AM‑1241 activates the CB₂ receptor with nanomolar affinity (K_i = 7.1 nM) and demonstrates >80‑fold selectivity over CB₁. This profile supports its use in dissecting CB₂‑specific pharmacological pathways.

References : Malan T. P Jr. et al.: Pain, 93(3), 239-45, 2001; Nackley A. G. et al.: Neuroscience, 119(3), 747-57, 2003; Yao B. B. et al.: Br. J.Pharmacol., 149(2), 145-54, 2006; Ibrahim M. M. et al.: Proc Natl Acad Sci., U S A., 100(18), 10529-33, 2003.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.