Apabetalone

SI-5595

Apabetalone, >98% (HPLC)

CAS No. : [1044870-39-4]

MDL No. : MFCD18633270

Synonyms : RVX000222; RVX-208

IUPAC Name : 2-(4-(2-Hydroxyethoxy)-3,5-dimethylphenyl)-5,7-dimethoxyquinazolin-4(3H)-one

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
100MG	Request A Quote		In Stock	Estimated to ship on 20 September 2026
250MG	Request A Quote		In Stock	Estimated to ship on 20 September 2026
1G	Request A Quote		In Stock	Estimated to ship on 20 September 2026
5G	Request A Quote		In Stock	Estimated to ship on 20 September 2026
10G	Request A Quote		In Stock	Estimated to ship on 20 September 2026

Applications : Apabetalone is an inhibitor of BET transcriptional regulators with selectivity for the second bromodomain. Apabetalone is being developed for the treatment of atherosclerosis and associated cardiovascular disease (CVD).

References : Picaud S. et al.: Proc Natl Acad Sci U S A. 110(49), 19754-9, 2013; McLure K. G. et al.: PLoS One 8(12), e83190, 2013; Jahagirdar R. et al.: Atherosclerosis 236(1), 91-100, 2014.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.