AR antagonist 5

SI-7506

AR antagonist 5, >98% (HPLC)

CAS No. : [2902679-53-0]

IUPAC Name : (2S)-N-(6-Cyano-5-(trifluoromethyl)pyridin-3-yl)-3-(6-(4-cyanophenyl)-3,6-diazabicyclo[3.1.1]heptan-3-yl)-2-hydroxy-2-methylpropanamide

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
250MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
500MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : This is a selective androgen receptor inhibitor with an IC₅₀ of 134.8 nM. It shows favorable pharmacokinetics, characterized by high skin exposure and low systemic (plasma) exposure, making it well‑suited for topical applications where localized AR blockade is desired without significant systemic activity.

References : Zhang W. et al.: J. Med. Chem., 67(1), 322-348, 2024.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.