ARD-2128

SI-7340

ARD-2128, >98% (HPLC)

CAS No. : [2222111-87-5]

IUPAC Name : N-((1r,3r)-3-(3-Chloro-4-cyanophenoxy)-2,2,4,4-tetramethylcyclobutyl)-4-(4-((1-(2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-5-yl)piperidin-4-yl)methyl)piperazin-1-yl)benzamide

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
5MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
10MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : ARD‑2128 functions as a high‑potency, orally bioavailable AR‑directed PROTAC that drives efficient AR degradation and downregulation of AR‑regulated genes in vivo. Its ability to inhibit tumor growth without detectable toxicity underscores its value as a tool compound for investigating AR‑driven prostate cancer biology.

References : Han X. et al.: J. Med. Chem., 64(17), 12831-12854, 2021.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.