AZ‑DprE1 inhibitor

SI-6069

AZ‑DprE1 inhibitor, >98% (HPLC)

IUPAC Name : N-(2-Fluoroethyl)-1-((6-methoxy-5-methylpyrimidin-4-yl)methyl)-1H-pyrrolo[3,2-b]pyridine-3-carboxamide

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
5MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
10MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : This is a potent AZ‑DprE1 inhibitor from the hydantoin‑replacement series targeting DprE1, an essential enzyme in Mycobacterium tuberculosis. This scaffold shows nanomolar biochemical affinity, strong cellular potency, and favorable physicochemical properties, positioning it as a promising noncovalent antituberculosis lead within the AZ‑DprE1 inhibitor class.

References : Balabon O. et al.: J. Med. Chem., 63(10), 5367-5386, 2020.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.