Azelaprag

SI-6240

Azelaprag, >98% (HPLC)

CAS No. : [2049980-18-7]

Synonyms : AMG-986

IUPAC Name : (2S,3R)-N-(4-(2,6-Dimethoxyphenyl)-5-(5-methylpyridin-3-yl)-4H-1,2,4-triazol-3-yl)-3-(5-methylpyrimidin-2-yl)butane-2-sulfonamide

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
5MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
10MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : Azelaprag is a sub‑nanomolar apelin receptor agonist (EC₅₀ = 0.32 nM) and represents a promising active molecule for modulating APJ‑dependent signaling. Its potency positions it as a valuable tool for studying apelin biology and related therapeutic mechanisms.

References : Ason B. et.al.: JCI Insight, 5(8), e132898, 2020.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.