BIIB-068

SI-6905

BIIB-068, >98% (HPLC)

CAS No. : [1798787-27-5]

IUPAC Name : 3-Isopropoxy-N-(2-methyl-4-(2-((1-methyl-1H-pyrazol-4-yl)amino)pyrimidin-4-yl)benzyl)azetidine-1-carboxamide

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
5MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
10MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : BIIB-068 reversibly inhibits BTK with strong potency (IC₅₀ = 1 nM; Kd = 0.3 nM) and displays >400‑fold selectivity relative to other kinases. Its oral activity and selectivity profile support its use in preclinical studies of autoimmune‑disease mechanisms involving BTK signaling.

References : Bin M. et al.: J. Med. Chem., 63(21), 12526-12541, 2020.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.