Birabresib

SI-6022

Birabresib, >98% (HPLC)

CAS No. : [202590-98-5]

MDL No. : MFCD26960949

Synonyms : MK-8628; OTX-015

IUPAC Name : (S)-2-(4-(4-Chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)-N-(4-hydroxyphenyl)acetamide

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
10MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
250MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
500MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
1G	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : Birabresib is a potent bromodomain (BRD2/3/4) inhibitor, exerts anti-tumor activity in triple-negative breast cancer models as single agent and in combination with everolimus.

References : Noel K. J. et al.: Mol Cancer Ther., 12(11_Supplement), C244, 2013;Marie-Magdelaine Coude M-M. et al.: Oncotarget., 6(19), 17698–17712, 2015; Lu P. et al.: Sci Rep., 6, 24100, 2016; Vazquez R. et al.: Oncotarget., 8(5), 7598-7613, 2017.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.