BMS-817399

SI-6605

BMS-817399, >98% (HPLC)

CAS No. : [1202400-18-7]

IUPAC Name : 1-((R)-1-((S)-4-(4-Chlorophenyl)-4-hydroxy-3,3-dimethylpiperidin-1-yl)-3-methyl-1-oxobutan-2-yl)-3-(2-hydroxy-2-methylpropyl)urea

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
5MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
10MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : BMS‑817399 is an orally active CCR1 antagonist that blocks receptor binding (IC₅₀ = 1 nM) and chemotaxis signaling (IC₅₀ = 6 nM). Its high potency and selectivity make it a valuable tool for probing CCR1‑driven inflammatory pathways, particularly in rheumatoid arthritis models.

References : Santella J. B. et al.: J. Med. Chem., 57(18), 7550-7564, 2014.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.