BMS-820132

SI-7716

BMS-820132, >98% (HPLC)

CAS No. : [1001419-18-6]

IUPAC Name : Diethyl ((3-(3-((5-(azetidine-1-carbonyl)pyrazin-2-yl)oxy)-5-isopropoxybenzamido)-1H-pyrazol-1-yl)methyl)phosphonate

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
250MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
500MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : BMS‑820132 partially activates glucokinase with high potency (AC₅₀= 29 nM) and lowers glucose levels in OGTT studies in normal, but not ZDF, rats. Its strong GK‑activating profile is associated with pharmacological toxicity.

References : Shi Y. et al.: J. Med. Chem., 65(5), 4291-4317, 2022.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.