Canertinib

SI-2481

Canertinib, >98% (HPLC)

CAS No. : [267243-28-7]

MDL No. : MFCD09837878

Synonyms : CI-1033; PD-183805

IUPAC Name : N-(4-((3-Chloro-4-fluorophenyl)amino)-7-(3-morpholinopropoxy)quinazolin-6-yl)acrylamide

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
10MG	55.00		Back Order	Estimated to ship on 04 October 2026
50MG	85.00		Back Order	Estimated to ship on 04 October 2026
100MG	125.00		Back Order	Estimated to ship on 04 October 2026
250MG	255.00		Back Order	Estimated to ship on 04 October 2026
500MG	455.00		Back Order	Estimated to ship on 04 October 2026

Applications : A potent, irreversible, orally available pan-ErbB inhibitor for EGFR and ErbB2 with IC₅₀ of 7.5 nM and 9.0 nM in autophosphorylation assay.

References : Smaill J. B. et al.: J. Med Chem., 43(7), 1380-1397, 2000; Erlichman C. et al.: Cancer Res., 61(2), 739-748, 2001; Nyati M. K. et al.: Clin Cancer Res., 10(2), 691-700, 2004; Slichenmyer W. J. et al.: Semin Oncol., 28 (5 Suppl 16), 80-85, 2001.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.