CCG-258747

SI-7892

CCG-258747, >98% (HPLC)

CAS No. : [2615910-00-2]

IUPAC Name : N-((1H-Indazol-3-yl)methyl)-5-((3S,4R)-3-((benzo[d][1,3]dioxol-5-yloxy)methyl)piperidin-4-yl)-2-fluorobenzamide

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
5MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
10MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : CCG-258747 is a selective GRK2 inhibitor (IC₅₀ = 18 nM) that modulates MOR internalization, IgE‑mediated anaphylaxis, and mast‑cell activation, supporting research into GRK2‑related diseases.

References : Bouley A. R. et al.: Mol Pharmacol., 97(6), 392-401, 2020; Thapaliya M. et al.: Front Immunol., 13, 1032497, 2022.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.