CCG-50014

SI-7706

CCG-50014, >98% (HPLC)

CAS No. : [883050-24-6]

IUPAC Name : 4-(4-Fluorobenzyl)-2-(p-tolyl)-1,2,4-thiadiazolidine-3,5-dione

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
5MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
10MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : CCG‑50014 selectively inhibits RGS4 (IC₅₀ = 30 nM; >20‑fold selectivity) by covalently binding two cysteines in an allosteric regulatory site. This covalent engagement translates into reduced nociceptive responses and enhanced opioid‑mediated analgesic effects in mouse formalin pain models.

References : Blazer L. L. et al.: Biochemistry, 50(15), 3181-92, 2011; Yoon S. Y. et al.: Anesth Analg., 120(3), 671-7, 2015.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.