Cebranopadol

SI-7709

Cebranopadol, >98% (HPLC)

CAS No. : [863513-91-1]

Synonyms : GRT-6005

IUPAC Name : (1r,4r)-6'-Fluoro-N,N-dimethyl-4-phenyl-4',9'-dihydro-3'H-spiro[cyclohexane-1,1'-pyrano[3,4-b]indol]-4-amine

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
5MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
10MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : Cebranopadol engages both the NOP and μ‑opioid receptors with high potency (K_i/EC₅₀ = 0.9/13 nM for NOP; 0.7/1.2 nM for MOR), producing a dual‑mechanism analgesic profile.

References : Linz K. et al.: J. Pharmacol. Exp. Ther., 349(3), 535-48, 2014; Schunk S. et al.: ACS Med. Chem. Lett., 5(8), 857-62, 2014.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.