Ceralasertib formate

SI-7574

Ceralasertib formate, >98% (HPLC)

CAS No. : [1352280-98-8]

Synonyms : AZD-6738 formate

IUPAC Name : (R)-Imino(methyl)(1-(6-((R)-3-methylmorpholino)-2-(1H-pyrrolo[2,3-b]pyridin-4-yl)pyrimidin-4-yl)cyclopropyl)-λ6-sulfanone formate

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
250MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
500MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : Ceralasertib formate potently inhibits ATR with a biochemical IC₅₀ of 1 nM and triggers downstream consequences of ATR blockade, including reduced cell viability, enhanced DNA damage, and induction of senescence. It shows clear antitumor efficacy in preclinical models.

References : Vendetti F. P. et al.: Oncotarget, 6(42), 44289-305, 2015; Kim H. J. et al.: Int. J. Cancer., 140(1), 109-119, 2017.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.