Derazantinib dihydrochloride

SI-7983

Derazantinib dihydrochloride, >98% (HPLC)

CAS No. : [1821329-75-2]

Synonyms : ARQ-087 dihydrochloride

IUPAC Name : (R)-6-(2-Fluorophenyl)-N-(3-(2-((2-methoxyethyl)amino)ethyl)phenyl)-5,6-dihydrobenzo[h]quinazolin-2-amine dihydrochloride

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
250MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
500MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : Derazantinib dihydrochloride is an orally active FGFR inhibitor that binds competitively to the ATP site, showing highest potency toward FGFR2. It suppresses FGFR phosphorylation and inhibits tumor growth in xenograft studies, making it a valuable tool for investigating FGFR‑dependent cancers.

References : Hall T. G. et al.: PLoS One, 11(9), e0162594, 2016; Balek L. et al.: Bone, 105, 57-66, 2017.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.