Dizocilpine maleate

SI-7703

Dizocilpine maleate, >98% (HPLC)

CAS No. : [77086-22-7]

Synonyms : (+)-MK-801 maleate

IUPAC Name : (5S,10R)-5-Methyl-10,11-dihydro-5H-5,10-epiminodibenzo[a,d][7]annulene maleate

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25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
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Applications : Dizocilpine maleate potently and selectively inhibits NMDA receptors through non‑competitive channel blockade, with a Kd of 37.2 nM in rat brain membranes. The maleate salt form is widely used in neuropharmacology and excitotoxicity research.

References : Wong E. H. et al.: Proc. Natl. Acad. Sci. U S A, 83(18), 7104-8, 1986; Wegener N. et al.: Neurosci. Lett., 503(1), 68-72, 2011; Huettner J. E. et al.: Proc. Natl. Acad. Sci. U S A, 85(4), 1307-11, 1988. Thomas D. M. et al.: Brain Res., 1050(1-2), 190-8, 2005; Brown T. E. et al.: Learn. Mem, 15(12), 857-65, 2008; Iijima Y. et al.:Nihon Shinkei Seishin Yakurigaku Zasshi. 16(1), 11-8, 1996.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.