Entospletinib

SI-6312

Entospletinib, >98% (HPLC)

CAS No. : [1229208-44-9]

Synonyms : GS-9973

IUPAC Name : 6-(1H-Indazol-6-yl)-N-(4-morpholinophenyl)imidazo[1,2-a]pyrazin-8-amine

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
10MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
250MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
500MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : Entospletinib is a potent, selective Syk inhibitor (IC₅₀ = 7.7 nM) with good oral bioavailability, making it a valuable tool for probing Syk‑mediated immune and inflammatory responses.

References : Currie K. S. et al.: J. Med. Chem., 57(9), 3856-73, 2014; Burke R. T. et al.: Oncotarget., 5(4), 908-15, 2014.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.