Fulvestrant

SL-9484

Fulvestrant, >98%

CAS No. : [129453-61-8]

Synonyms : ICI 182780; ZD 9238; ZM 182780

IUPAC Name : (7R,8R,9S,13S,14S,17S)-13-Methyl-7-(9-((4,4,5,5,5-pentafluoropentyl)sulfinyl)nonyl)-7,8,9,11,12,13,14,15,16,17-decahydro-6H-cyclopenta[a]phenanthrene-3,17-diol

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
250MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
500MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : Fulvestrant is a pure antiestrogen and a potent estrogen receptor (ER) antagonist with an IC50 of 9.4 nM. It is also a GPR30 agonist. Fulvestrant effectively inhibits the growth of ER-positive MCF-7 cells with an IC50 of 0.29 nM. It also induces autophagy and has antitumor efficacy.

References : Wakeling A. E. et al.: Cancer Res., 51(15), 3867-73, 1991; Yu X. et al.: Mol Cancer 14, 208, 2015; Osborne C. K. et al.: Br. J. Cancer 90 Suppl 1, S2-6, 2004; Garner F. et al.: Anticancer Drugs 26(9), 948-56, 2015; Julia K. et al.: Eur. J. Neurosci., 27(7), 1700-9, 2008.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.