Futibatinib

SI-6731

Futibatinib, >98% (HPLC)

CAS No. : [1448169-71-8]

Synonyms : TAS-120

IUPAC Name : (S)-1-(3-(4-Amino-3-((3,5-dimethoxyphenyl)ethynyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)pyrrolidin-1-yl)prop-2-en-1-one

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
5MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
10MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : Futibatinib is an irreversible FGFR inhibitor with low‑nanomolar potency across FGFR1–4. It retains robust inhibitory activity against wild‑type FGFR2 and key FGFR2 resistance mutations (V565I, N550H, E566G), making it valuable for studying FGFR‑driven tumor biology and acquired resistance.

References : Goyal L. et al.: Cancer Discov., 9(8), 1064-1079, 2019; Kalyukina M. et al.: Chem. Med. Chem., 14(4), 494-500, 2019; Lamarca A. et al.: J. Hepatol., S0168, 8278(20)30165-3, 2020.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.