Galeflaprit fumarate

SI-8152

Galeflaprit fumarate, >98% (HPLC)

CAS No. : [3026790-19-9]

Synonyms : LXE-408 fumarate

IUPAC Name : N-(4-Fluoro-3-(6-(3-methylpyridin-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl)phenyl)-2,4-dimethyloxazole-5-carboxamide maleate

Price And Availability
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25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
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Applications : Galeflaprit fumarate selectively inhibits the kinetoplastid proteasome in a non‑competitive manner, with strong potency against L. donovani (IC₅₀/EC₅₀ = 0.04 µM). Its low propensity to cross the blood–brain barrier supports its suitability for visceral leishmaniasis research and development.

References : Nagle A. et al.: J. Med. Chem., 63(19), 10773-10781, 2020.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.