GCN2-IN-7

SI-7176

GCN2-IN-7, >98% (HPLC)

CAS No. : [2396465-33-9]

IUPAC Name : (1R,3R)-3-((3-Bromo-1-(4-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl)-1H-pyrazolo[3,4-d]pyrimidin-6-yl)amino)-N,1-dimethylcyclopentane-1-carboxamide

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
5MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
10MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : GCN2‑IN‑7 is an orally active and selective GCN2 inhibitor with IC₅₀ = 5 nM. It demonstrates in vivo anti‑tumor activity, making it a useful tool compound for studying GCN2‑dependent stress signaling and its role in cancer biology.

References : Jackson J. J. et al.: J. Med. Chem., 65(19), 12895-12924, 2022.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.