Gedatolisib

SI-1783

Gedatolisib, 98% (HPLC)

CAS No. : [1197160-78-3]

MDL No. : MFCD16875679

Synonyms : PF-05212384, PKI-587

IUPAC Name : 1-(4-(4-(Dimethylamino)piperidine-1-carbonyl)phenyl)-3-(4-(4,6-dimorpholino-1,3,5-triazin-2-yl)phenyl)urea

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
5MG	160.00		Back Order	Estimated to ship on 04 October 2026
10MG	250.00		Back Order	Estimated to ship on 04 October 2026
25MG	350.00		Back Order	Estimated to ship on 04 October 2026
50MG	650.00		Back Order	Estimated to ship on 04 October 2026
100MG	950.00		Back Order	Estimated to ship on 04 October 2026

Applications : Gedatolisib is a highly potent dual inhibitor of PI3Kα, PI3Kγ and mTOR with IC₅₀ of 0.4 nM, 5.4 nM and 1.6 nM in cell-free assays, respectively.

References : Venkatesan A. M. et al. J. Med. Chem., 53(6), 2636-2645, 2010; Mallon R. et al.: Clin. Cancer Res.,17(10), 3193-203, 2011; Gedaly R. et al.: J. Surg. Res., 185(1), 225-230, 2013; D'Amato V. et al.: Br. J. Cancer 110(12), 2887-95, 2014.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.