GPR84 antagonist 3

SI-7139

GPR84 antagonist 3, >98% (HPLC)

CAS No. : [2815263-05-7]

IUPAC Name : 4-(4-(3-((1H-Indol-3-yl)methyl)-5-phenyl-1,2,4-triazin-6-yl)benzyl)morpholine

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
5MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
10MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : This is a potent GPR84 antagonist that inhibits GTPγS binding with a pIC₅₀ of 8.28, indicating strong nanomolar activity. It demonstrates a favorable pharmacokinetic profile, making it suitable for in vivo studies of GPR84‑mediated inflammatory signaling and related disease models.

References : Mahindra A. et al.: J. Med. Chem., 65(16), 11270-11290, 2022.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.