GSK-1904529A

SI-6396

GSK-1904529A, >98% (HPLC)

CAS No. : [1089283-49-7]

IUPAC Name : N-(2,6-Difluorophenyl)-5-(3-(2-((5-ethyl-2-methoxy-4-(4-(4-(methylsulfonyl)piperazin-1-yl)piperidin-1-yl)phenyl)amino)pyrimidin-4-yl)imidazo[1,2-a]pyridin-2-yl)-2-methoxybenzamide

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
5MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
10MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : GSK-1904529A selectively inhibits IGF‑1R and IR with low‑nanomolar potency through ATP‑competitive binding while showing negligible activity across a broad kinase panel. This selectivity translates into robust anti‑tumor effects in preclinical models of IGF‑1R/IR‑dependent cancers.

References : Sabbatini P. et al.: Clin. Cancer Res., 15(9), 3058-3067, 2009; Zhou Q. et al.: Mol. Med. Rep., 12(3), 3381-3385, 2015.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.