GSK-217

SI-6225

GSK-217, >98% (HPLC)

CAS No. : [2748687-92-3]

IUPAC Name : 2-((1H-Indol-4-yl)methyl)-N-ethyl-6-(1-methyl-1H-1,2,3-triazol-4-yl)isonicotinamide

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
250MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
500MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : GSK-217 selectively targets the BD2 domains of BET proteins and exhibits high solubility and strong biochemical potency. It is a valuable tool compound for investigating BD2‑dependent transcriptional programs in cancer biology and immune‑inflammation research.

References : Aylott H. E. et al.: J. Med. Chem., 64(6), 3249-3281, 2021.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.