GSK-2816126A

SI-6180

GSK-2816126A, >98% (HPLC)

CAS No. : [1346574-57-9]

Synonyms : GSK-126

IUPAC Name : (S)-1-(Sec-butyl)-N-((4,6-dimethyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-3-methyl-6-(6-(piperazin-1-yl)pyridin-3-yl)-1H-indole-4-carboxamide

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
250MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
500MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : GSK-2816126A is a selective EZH2 inhibitor with nanomolar potency (IC₅₀ = 9.9 nM) that blocks PRC2‑driven histone H3K27 methylation. It serves as a key tool compound for studying EZH2‑regulated transcriptional programs.

References : McCabe M. T. et al.: Nature, 492(7427), 108-12, 2012; Sato T. et al.: Sci. Rep., 3, 1911, 2013.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.