GSK-2981278

SI-6849

GSK-2981278, >98% (HPLC)

CAS No. : [1474110-21-8]

IUPAC Name : N-(4-Ethylphenyl)-3-(hydroxymethyl)-N-isobutyl-4-((tetrahydro-2H-pyran-4-yl)methoxy)benzenesulfonamide

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
5MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
10MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : GSK-2981278 selectively targets RORγ as a potent inverse agonist, blocking IL‑17 promoter activation and impairing RORγ binding to DNA. Its strong mechanistic activity supports its use in studies of Th17‑driven immune signaling.

References : Smith S. H. et al.: 11(2); e0147979, 2016.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.