GW-501516

SI-7334

GW-501516, >98% (HPLC)

CAS No. : [317318-70-0]

Synonyms : GW-1516; GSK-516

IUPAC Name : 2-(2-Methyl-4-(((4-methyl-2-(4-(trifluoromethyl)phenyl)thiazol-5-yl)methyl)thio)phenoxy)acetic acid

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
250MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
500MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : GW-501516 activates PPARδ with nanomolar potency (EC₅₀ = 1.1 nM), supporting its use in studies of lipid metabolism, energy homeostasis, and PPARδ‑dependent transcriptional regulation.

References : Wei Z. L. et al.: J. Org Chem., 68(23), 9116-8, 2003; Mosti M. P. et al.: Endocrinology, 155(6), 2178-89, 2014; Yang X. et al.: PLoS One, 6(9), e25271, 2011; Chen W. et al.: Sci Rep., 5, 9884, 2015; Ji Y. et al.: Front Pharmacol, 9, 648, 2018.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.