IBET-567

SI-6928

IBET-567, >98% (HPLC)

CAS No. : [1887237-54-8]

IUPAC Name : (2S,4R)-1-Acetyl-4-((5-chloropyrimidin-2-yl)amino)-2-methyl-1,2,3,4-tetrahydroquinoline-6-carboxamide

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
5MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
10MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : I‑BET567 potently targets BET bromodomains, with high affinity for BRD4 BD1 and BD2, and displays oral activity. It has demonstrated significant antitumor and anti‑inflammatory effects in mouse models, highlighting its relevance for studying BET‑dependent transcriptional programs.

References :
Humphreys P. G. et al.: J. Med. Chem., 65(3), 2262-2287, 2022.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.