IIIM-290

SI-7805

IIIM-290, >98% (HPLC)

CAS No. : [2213468-64-3]

IUPAC Name : 2-((E)-2,6-Dichlorostyryl)-5,7-dihydroxy-8-((3R,4S)-3-hydroxy-1-methylpiperidin-4-yl)-4H-chromen-4-one

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
250MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
500MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : IIIM‑290 potently inhibits CDK2 and CDK9 with IC₅₀ values of 90 nM and 94 nM, respectively. As an orally active compound, it serves as a useful tool for probing CDK‑dependent pathways involved in cell‑cycle progression and transcriptional regulation.

References : Bharate S. B. et al.: J. Med. Chem., 61(4), 1664-1687, 2018.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.