Itraconazole

SL-7753

Itraconazole, >98%

CAS No. : [84625-61-6]

Synonyms : Oriconazole; R-51211; Sporamelt; Sporanox; Triasporin; Itrizole

IUPAC Name : 4-(4-(4-(4-(((2R,4S)-2-((1H-1,2,4-Triazol-1-yl)methyl)-2-(2,4-dichlorophenyl)-1,3-dioxolan-4-yl)methoxy)phenyl)piperazin-1-yl)phenyl)-2-(sec-butyl)-2,4-dihydro-3H-1,2,4-triazol-3-one

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
1G	10.00		In Stock	Estimated to ship on 20 September 2026
5G	29.00		In Stock	Estimated to ship on 20 September 2026
10G	50.00		In Stock	Estimated to ship on 20 September 2026
25G	95.00		In Stock	Estimated to ship on 20 September 2026
100G	295.00		In Stock	Estimated to ship on 20 September 2026
500G	995.00		In Stock	Estimated to ship on 20 September 2026

Applications : Itraconazole is a relatively potent inhibitor of CYP3A4 with IC₅₀ of 6.1 nM, used as a triazole antifungal agent. Itraconazole is a potent antagonist of the Hedgehog (Hh) signaling pathway.

References : Isoherranen N. et al. Drug Metab Dispos, 32(10), 1121-1131, 2004; Kim J. et al. Cancer Cell., 17(4), 388-399, 2010; Oakley K. L. et al. Antimicrob Agents Chemother., 41(5), 1124-1126, 1997; Zuckerman J. M. et al. Infect Control Hosp Epidemiol., 15(6), 397-410, 1994; Leyden J. et al. J. Am Acad Dermatol, 38(5 Pt 3), S42-47, 1998; Isoherranen N. et al. Drug Metab Dispos., 32(10):1121-31, 2004.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.