Lenumlostat

SI-6117

Lenumlostat, >98% (HPLC)

CAS No. : [2007885-39-2]

Synonyms : PAT-1251; GB-2064

IUPAC Name : (3-((4-(Aminomethyl)-6-(trifluoromethyl)pyridin-2-yl)oxy)phenyl)((3R,4R)-3-fluoro-4-hydroxypyrrolidin-1-yl)methanone

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
5MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
10MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
250MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
500MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : PAT‑1251 potently inhibits LOXL2 (hLOXL2 IC₅₀ = 0.71 µM) and shows activity against hLOXL3, as well as LOXL2 from multiple species. With strong oral bioactivity and selectivity, it is a valuable tool for investigating LOXL2‑driven fibrotic pathways in diverse animal models.

References : Rowbottom M. W. et al.: J. Med. Chem., 60(10), 4403-4423, 2017.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.