Lenumlostat hydrochloride

SI-6118

Lenumlostat hydrochloride, >98% (HPLC)

CAS No. : [2098884-53-6]

Synonyms : PAT-1251 hydrochloride; GB-2064 hydrochloride

IUPAC Name : (3-((4-(Aminomethyl)-6-(trifluoromethyl)pyridin-2-yl)oxy)phenyl)((3R,4R)-3-fluoro-4-hydroxypyrrolidin-1-yl)methanone hydrochloride

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
250MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
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Applications : PAT‑1251 hydrochloride selectively inhibits LOXL2 (hLOXL2 IC₅₀ = 0.71 µM) and shows activity against hLOXL3, as well as LOXL2 from multiple species. With strong oral activity and cross‑species potency, it is a valuable tool for probing LOXL2‑driven fibrotic pathways in diverse experimental models.

References : Rowbottom M. W. et al.: J. Med. Chem., 60(10), 4403-4423, 2017.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.