lunresertib

SI-7485

lunresertib, >98% (HPLC)

CAS No. : [2719793-90-3]

Synonyms : RP-6306

IUPAC Name : 2-Amino-1-(3-hydroxy-2,6-dimethylphenyl)-5,6-dimethyl-1H-pyrrolo[2,3-b]pyridine-3-carboxamide

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
5MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
10MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : Lunresertib selectively inhibits PKMYT1 with an IC₅₀ of 14 nM and displays minimal off‑target kinase binding. Its mechanism disrupts PKMYT1‑mediated cell‑cycle progression, resulting in pronounced anticancer activity.

References : Szychowski J. et al.: J. Med.Chem., 65(15), 10251-10284, 2022; Gallo D. et al.: Nature, 604(7907), 749-756, 2022.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.