Molibresib carboxylic acid

SI-5982

Molibresib carboxylic acid, >98% (HPLC)

CAS No. : [1300019-38-8]

Synonyms : GSK525762A carboxylic acid; Deasethyl molibresib

IUPAC Name : 2-((4S)-6-(4-Chlorophenyl)-8-methoxy-1-methyl-4H-benzo[f][1,2,4]triazolo[4,3-a][1,4]diazepin-4-yl)acetic acid; I-BET762 carboxylic acid

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
5MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
10MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
250MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
500MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : Molibresib carboxylic acid is an I-BET-762-based warhead ligand for conjugation reactions of PROTAC targeting on BET. Molibresib carboxylic acid is a BRD4 inhibitor.

References : Mirguet O. et al.: J. Med Chem., 56(19), 7501-15, 2013.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.