MRTX-9768

SI-8104

MRTX-9768, >98% (HPLC)

CAS No. : [2629314-68-5]

IUPAC Name : 2-(4-(4-(Aminomethyl)-1-oxo-1,2-dihydrophthalazin-6-yl)-1-methyl-1H-pyrazol-5-yl)-3-fluoro-1-naphthonitrile

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
5MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
10MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : MRTX-9768 is an orally active, first‑in‑class PRMT5–MTA complex inhibitor with strong potency and selectivity. By exploiting MTA‑dependent PRMT5 engagement, it provides a targeted approach for studying PRMT5‑driven malignancies.

References : Christopher R. et al.: Cancer Res., 81(13 Suppl), 2021; Chen Y. et al.: Biomed. Pharmacother., 144, 112252, 2021.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.