Oliceridine

SI-7633

Oliceridine, >98% (HPLC)

CAS No. : [1401028-24-7]

Synonyms : Olinvo, TRV-130

IUPAC Name : (R)-N-((3-Methoxythiophen-2-yl)methyl)-2-(9-(pyridin-2-yl)-6-oxaspiro[4.5]decan-9-yl)ethan-1-amine

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
5MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
10MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : Oliceridine selectively activates the μ‑opioid receptor with strong G‑protein bias and high potency (pEC₅₀ = 8.1). Its signaling profile distinguishes it from conventional opioids and makes it valuable for probing biased MOR‑mediated analgesia.

References : Chen X. T. et al.: J. Med. Chem., 56(20), 8019-31, 2013; DeWire S. M. et al.: J. Pharmacol. Exp. Ther., 344(3), 708-17, 2013; Schneider S. et al.: Biochemistry, 55(46), 6456-6466, 2016.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.