PF-04217903 phenolsulfonate

SI-8043

PF-04217903 phenolsulfonate, >98% (HPLC)

CAS No. : [1159490-85-3]

IUPAC Name : 2-(4-(1-(Quinolin-6-ylmethyl)-1H-[1,2,3]triazolo[4,5-b]pyrazin-6-yl)-1H-pyrazol-1-yl)ethan-1-ol 4-hydroxybenzenesulfonate

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
250MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
500MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : PF‑04217903 phenolsulfonate is a highly potent ATP‑competitive c‑MET inhibitor (K_i= 4.8 nM) with exceptional selectivity, exceeding 1,000‑fold over 208 kinases tested. It effectively blocks MET‑regulated signaling pathways and displays antiangiogenic activity, making it a valuable tool for investigating MET‑mediated tumor biology.

References : Zou H. Y. et al.: Mol. Cancer Ther., 11(4), 1036-47, 2012; Cui J. J. et al.: J. Med. Chem., 55(18), 8091-109, 2012; Timofeevski S. L. et al.: Biochemistry, 48(23), 5339-49, 2009.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.