Pictilisib

SI-1785

Pictilisib, 98% (HPLC)

CAS No. : [957054-30-7]

MDL No. : MFCD11616196

Synonyms : GDC-0941

IUPAC Name : 4-(2-(1H-Indazol-4-yl)-6-((4-(methylsulfonyl)piperazin-1-yl)methyl)thieno[3,2-d]pyrimidin-4-yl)morpholine

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
5MG	95.00		Back Order	Estimated to ship on 04 October 2026
10MG	155.00		Back Order	Estimated to ship on 04 October 2026
25MG	255.00		Back Order	Estimated to ship on 04 October 2026
50MG	355.00		Back Order	Estimated to ship on 04 October 2026
100MG	555.00		Back Order	Estimated to ship on 04 October 2026
250MG	955.00		Back Order	Estimated to ship on 04 October 2026

Applications : Pictilisib is a potent inhibitor of PI3Kα/δ with IC₅₀ of 3 nM in cell-free assays, with modest selectivity against p110β (11-fold) and p110γ (25-fold).

References : Wallin J. J. et al.: Clin Cancer Res., 18(14), 3901-3911, 2012; Folkes A. J. et al.: J. Med. Chem., 51(18), 5522-5532, 2008; Cheng H. et al.: Cancer Res., 74(1), 15-23, 2014.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.