rac-AMC-487

SI-7155

rac-AMC-487, >98% (HPLC)

CAS No. : [947536-03-0]

Synonyms : (±)-AMG-487

IUPAC Name : N-(1-(3-(4-Ethoxyphenyl)-4-oxo-3,4-dihydropyrido[2,3-d]pyrimidin-2-yl)ethyl)-N-(pyridin-3-ylmethyl)-2-(4-(trifluoromethoxy)phenyl)acetamide

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
5MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
10MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : (±)-AMG-487 is the racemic mixture of AMG-487, an orally active and selective CXCR3 antagonist that inhibits CXCL10 and CXCL11 binding with IC₅₀ values of 8.0 and 8.2 nM, respectively.

References : Johnson M. et al.: Bioorg.Med. Chem. Lett., 17(12), 3339-43, 2007.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.