Relcovaptan

SI-7479

Relcovaptan, >98% (HPLC)

CAS No. : [150375-75-0]

Synonyms : SR-49059

IUPAC Name : (S)-1-((2R,3S)-5-Chloro-3-(2-chlorophenyl)-1-((3,4-dimethoxyphenyl)sulfonyl)-3-hydroxyindoline-2-carbonyl)pyrrolidine-2-carboxamide

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
5MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
10MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : Relcovaptan selectively antagonizes the vasopressin V1a receptor with nanomolar affinity (K_i = 1.4 nM) and demonstrates oral activity. It is widely used to probe V1a‑dependent signaling in cardiovascular, endocrine, and stress‑related research.

References : Serradeil-Le Gal C. et al.: Am. J. Physiol., 268(1 Pt 2), H404-10, 1995; Shuaib A. et al.: Stroke, 33(12), 3033-7, 2022.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.