Rilzabrutinib

SI-6287

Rilzabrutinib, >98% (HPLC)

CAS No. : [1575596-29-0]

Synonyms : PRN-1008

IUPAC Name : (R,E)-2-(3-(4-Amino-3-(2-fluoro-4-phenoxyphenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)piperidine-1-carbonyl)-4-methyl-4-(4-(oxetan-3-yl)piperazin-1-yl)pent-2-enenitrile

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
5MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
10MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : Rilzabrutinib is a reversible covalent BTK inhibitor with high selectivity and low‑nanomolar potency (IC₅₀ = 1.3 nM), making it a valuable tool for probing BTK‑dependent pathways.

References : Smith P. F. et al.: Br. J. Clin. Pharmacol., 83(11), 2367-2376, 2017;Hill R. J. et al.: Annals of the Rheumatic Diseases, 74(Suppl 2), 216, 2015.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.