Rimegepant hemisulfate

SI-7637

Rimegepant hemisulfate, >98% (HPLC)

CAS No. : [1642783-82-1]

Synonyms : BMS-927711 hemisulfate; BHV-3000 hemisulfate

IUPAC Name : (5S,6S,9R)-5-Amino-6-(2,3-difluorophenyl)-6,7,8,9-tetrahydro-5H-cyclohepta[b]pyridin-9-yl 4-(2-oxo-2,3-dihydro-1H-imidazo[4,5-b]pyridin-1-yl)piperidine-1-carboxylate hemisulfate

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
250MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
500MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : Rimegepant hemisulfate selectively and competitively blocks the CGRP receptor with sub‑nanomolar affinity (K_i= 0.027 nM) and potent functional activity (IC₅₀= 0.14 nM). Its oral activity and strong receptor selectivity make it a valuable tool compound for migraine research.

References : Luo G. et al.: J. Med. Chem. 55(23), 10644-51, 2012.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.