Rimegepant sulfate hydrate

SI-7638

Rimegepant sulfate hydrate, >98% (HPLC)

CAS No. : [1374024-48-2]

Synonyms : BMS-927711 sulfate hydrate; BHV-3000 sulfate hydrate

IUPAC Name : (5S,6S,9R)-5-Amino-6-(2,3-difluorophenyl)-6,7,8,9-tetrahydro-5H-cyclohepta[b]pyridin-9-yl 4-(2-oxo-2,3-dihydro-1H-imidazo[4,5-b]pyridin-1-yl)piperidine-1-carboxylate sulfate hydrate

Price And Availability
Pack Size	Price in USD	Add To Shopping Cart	Availability	Shipping Status
5MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
10MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
25MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
50MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026
100MG	Request A Quote		Back Order	Estimated to ship on 04 October 2026

Applications : Rimegepant sulfate hydrate selectively blocks the CGRP receptor with sub‑nanomolar affinity (K_i = 0.027 nM) and potent functional activity (IC₅₀= 0.14 nM). Its oral activity and receptor selectivity make it a valuable tool compound for migraine research and CGRP‑pathway investigations.

References : Blair H. A.: CNS Drugs, 37(3), 255-265, 2023; Luo G. et al.: J. Med. Chem., 55(23), 10644-51, 2012.

Storage : Keep container tightly closed under nitrogen or argon and refrigerate for long-term shelf life.

Caution : In case of contact with skin or eyes, rinse immediately with plenty of water and seek medical advice. Wear suitable protective clothing and gloves.